IUPHAR/BPS Guide to Pharmacology CITE
https://doi.org/10.2218/gtopdb/F201/2023.3
SLC23 family of ascorbic acid transporters in GtoPdb v.2023.3
James M. May1
- Vanderbilt University, USA
Abstract
Predicted to be 12 TM segment proteins, members of this family transport the reduced form of ascorbic acid (while the oxidized form may be handled by members of the SLC2 family (GLUT1/SLC2A1, GLUT3/SLC2A3 and GLUT4/SLC2A4). phloretin is considered a non-selective inhibitor of these transporters, with an affinity in the micromolar range [1].
Contents
This is a citation summary for SLC23 family of ascorbic acid transporters in the
Guide to Pharmacology
database (GtoPdb). It exists purely as an adjunct to the database to
facilitate the recognition of citations to and from the database by
citation analyzers. Readers will almost certainly want to visit the
relevant sections of the database which are given here under database
links.
GtoPdb is an expert-driven
guide to pharmacological targets and the substances that act on them.
GtoPdb is a reference work which is most usefully represented as an
on-line database. As in any publication this work should be
appropriately cited, and the papers it cites should also be
recognized. This document provides a citation for the relevant parts
of the database, and also provides a reference list for the research
cited by those parts. For further details see [2].
Please note that the database version for the citations given in
GtoPdb are to the most recent preceding version
in which the family or its subfamilies and targets were substantially
changed. The links below are to the current version. If you
need to consult the cited version, rather than the most recent version, please contact
the GtoPdb curators.
Database links
SLC23 family of ascorbic acid transporters
https://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=201
Transporters
SVCT1(Sodium-dependent vitamin C transporter 1)
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1041
SVCT2(Sodium-dependent vitamin C transporter 2)
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1042
SVCT3(Sodium-dependent vitamin C transporter 3)
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1043
SNBT1(Sodium-dependent nucleobase transporter)
https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1044
References
- Alexander SPH, Kelly E, Mathie A, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Pawson AJ and Sharman JL et al.. (2019) THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Transporters. Br J Pharmacol 176 Suppl 1: S397-S493 [PMID:31710713]
- Buneman P, Christie G, Davies JA, Dimitrellou R, Harding SD, Pawson AJ, Sharman JL and Wu Y. (2020) Why data citation isn't working, and what to do about it Database 2020 [PMID:32367113]
- MacDonald L, Thumser AE and Sharp P. (2002) Decreased expression of the vitamin C transporter SVCT1 by ascorbic acid in a human intestinal epithelial cell line. Br J Nutr 87: 97-100 [PMID:11895172]
- Tsukaguchi H, Tokui T, Mackenzie B, Berger UV, Chen XZ, Wang Y, Brubaker RF and Hediger MA. (1999) A family of mammalian Na+-dependent L-ascorbic acid transporters. Nature 399: 70-5 [PMID:10331392]
- Yamamoto S, Inoue K, Murata T, Kamigaso S, Yasujima T, Maeda JY, Yoshida Y, Ohta KY and Yuasa H. (2010) Identification and functional characterization of the first nucleobase transporter in mammals: implication in the species difference in the intestinal absorption mechanism of nucleobases and their analogs between higher primates and other mammals. J Biol Chem 285: 6522-31 [PMID:20042597]