IUPHAR/BPS Guide to Pharmacology CITE
https://doi.org/10.2218/gtopdb/F39/2021.3

Melatonin receptors in GtoPdb v.2021.3



Daniel P. Cardinali1, Philippe Delagrange2, Margarita L. Dubocovich3, Ralf Jockers4, Diana N. Krause5, Regina Pekelmann Markus6, James Olcese7, Jesús Pintor8, Nicolas Renault9, David Sugden10, Gianluca Tosini11 and Darius Paul Zlotos12
  1. Pontificia Universidad Católica Argentina Buenos Aires, Argentina
  2. Servier, France
  3. University at Buffalo (SUNY), USA
  4. Université Paris Descartes, France
  5. University of California Irvine, USA
  6. University of São Paulo, Brazil
  7. Florida State University, USA
  8. Universidad Complutense de Madrid, Spain
  9. Université Lille 2, France
  10. King's College London, UK
  11. Morehouse School of Medicine, USA
  12. German University in Cairo, Egypt


Abstract

Melatonin receptors (nomenclature as agreed by the NC-IUPHAR Subcommittee on Melatonin Receptors [40]) are activated by the endogenous ligands melatonin and clinically used drugs like ramelteon, agomelatine and tasimelteon.

Contents

This is a citation summary for Melatonin receptors in the Guide to Pharmacology database (GtoPdb). It exists purely as an adjunct to the database to facilitate the recognition of citations to and from the database by citation analyzers. Readers will almost certainly want to visit the relevant sections of the database which are given here under database links.

GtoPdb is an expert-driven guide to pharmacological targets and the substances that act on them. GtoPdb is a reference work which is most usefully represented as an on-line database. As in any publication this work should be appropriately cited, and the papers it cites should also be recognized. This document provides a citation for the relevant parts of the database, and also provides a reference list for the research cited by those parts. For further details see [20].

Please note that the database version for the citations given in GtoPdb are to the most recent preceding version in which the family or its subfamilies and targets were substantially changed. The links below are to the current version. If you need to consult the cited version, rather than the most recent version, please contact the GtoPdb curators.

Database links

Melatonin receptors
https://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=39
Introduction to Melatonin receptors
https://www.guidetopharmacology.org/GRAC/FamilyIntroductionForward?familyId=39
    Receptors
            MT1 receptor
            https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=287
            MT2 receptor
            https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=288

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