IUPHAR/BPS Guide to Pharmacology CITE
https://doi.org/10.2218/gtopdb/F34/2020.4

Kisspeptin receptor (version 2020.4) in the IUPHAR/BPS Guide to Pharmacology Database



Anthony P. Davenport1, Janet J. Maguire1, Edward J. Mead1 and Adam J. Pawson2
  1. University of Cambridge, UK
  2. The University of Edinburgh, UK


Abstract

The kisspeptin receptor (nomenclature as agreed by the NC-IUPHAR Subcommittee on the kisspeptin receptor [9]), like neuropeptide FF (NPFF), prolactin-releasing peptide (PrP) and QRFP receptors (provisional nomenclature) responds to endogenous peptides with an arginine-phenylalanine-amide (RFamide) motif. kisspeptin-54 (KP54, originally named metastin), kisspeptin-13 (KP13) and kisspeptin-10 (KP10) are biologically-active peptides cleaved from the KISS1 (Q15726) gene product. Kisspeptins have roles in, for example, cancer metastasis, fertility/puberty regulation and glucose homeostasis.

Contents

This is a citation summary for Kisspeptin receptor in the Guide to Pharmacology database (GtoPdb). It exists purely as an adjunct to the database to facilitate the recognition of citations to and from the database by citation analyzers. Readers will almost certainly want to visit the relevant sections of the database which are given here under database links.

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Database links

Kisspeptin receptor
http://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=34
Introduction to Kisspeptin receptor
http://www.guidetopharmacology.org/GRAC/FamilyIntroductionForward?familyId=34
    Receptors
            kisspeptin receptor
            http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=266

References

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