IUPHAR/BPS Guide to Pharmacology CITE

Endothelin receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

Pedro D'Orléans-Juste1, Anthony P. Davenport2, Théophile Godfraind3, Janet J. Maguire2, Eliot H. Ohlstein4 and Robert R. Ruffolo5
  1. University of Sherbrooke, Canada
  2. University of Cambridge, UK
  3. Université Catholique de Louvain, Belgium
  4. Drexel University, USA
  5. Wyeth Pharmaceuticals, USA


Endothelin receptors (nomenclature as agreed by the NC-IUPHAR Subcommittee on Endothelin Receptors [24]) are activated by the endogenous 21 amino-acid peptides endothelins 1-3 (endothelin-1, endothelin-2 and endothelin-3).


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Database links

Endothelin receptors
Introduction to Endothelin receptors
            ETA receptor
            ETB receptor


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